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What is this drugs used for? and what could be the advese effect of that drug? D

ID: 167456 • Letter: W

Question

What is this drugs used for? and what could be the advese effect of that drug?

DRUG

MECHANISM OF ACTION

CLINICAL INDICATION (select one)

EXPECTED ADVERSE EFFECT (select one)

Donepizil (Aricept)

Acetylcholinesterase Inhibitor

Alzheimer's / Parkinson's / Schizophrenia

Urine retention / Bradycardia / Dystonic Reaction

Citalopam (Celexa)

SERT Inhibitor

Psychosis / Obsessive Compulsive / Parkinson's

SLUDGE / Serotonin Syndrome / Hypotension

Phenelzine (Nardil)

Nonselective MAO Inhibitor

Depression / Migraine Headache / Schizophrenia

Bradycardia / Hypertension / Sedation

Clobazam (Onfi)

GABA-A modulator

Analgesic / Anticonvulsant / Anxiolytic

Dystonic Reaction / Sedation / Bronchorrhea & Bronchospasm

Desvenlafaxine (Pristiq)

SNRI

Schizophrenia / Parkinson's / Antidepressant

Hypertension / Hypotension / Dystonic Reaction

Alprazolam (Xanax)

GABA-A modulator

Insomnia / Depression / Analgesic

Sedation / Constipation / Dystonic Reaction

Lisdexamfetamine (Vyvanse)

Degranulation of NE and DA vesicles

Alzheimer's / ADHD / Schizophrenia

Dystonic Reaction / Serotonin Syndrome / Tachycardia

Olanzapine (Zyprexa)

5HT2a Antagonist / D1 Antagonist

Psychosis / Antidepressant / Weight Loss

Serotonin Syndrome / Dystonic Reaction / SLUDGE

Zaleplon (Sonata)

nonbenzodiazepine GABA-A Agonist

Parkinson's / Analgesic / Insomnia

Bradycardia / Hypertension / Sedation

Selegeline (Anipryl)

MAO-B Selective Inhibition

Schizophrenia / Parkinson's / ADHD

Vomiting / Dystonic Reaction / Diarrhea & Salivation

Baclofen (Lioresal)

GABA-B Agonist

Insomnia / Anticonvulsant / Muscular Spasms

Seizures / Sedation / Tachycardia & Hypertension

Bupropion (Wellbutrin)

DAT and NET Inhibition

Depression / Insomnia / Schizophrenia

Tachycardia & Hypertension / SLUDGE / Sedation

Promethazine (Phenergan)

D1 D2 Antagonist

Analgesic / Antiemetic / Antidepressant

SLUDGE / Dystonic Reaction / Serotonin Syndrome

Paroxetine (Paxil)

SERT inhibition

ADHD / Parkinson's / Depression

Serotonin Syndrome / Dystonic Reaction / Hypotension

Ropinirole (Requip)

D2 Agonist

ADHD / Parkinson's / Depression

Nausea and Emesis / Bradycardia / Serotonin Syndrome

What is this drugs used for? and what could be the advese effect of that drug?

DRUG

MECHANISM OF ACTION

CLINICAL INDICATION (select one)

EXPECTED ADVERSE EFFECT (select one)

Donepizil (Aricept)

Acetylcholinesterase Inhibitor

Alzheimer's / Parkinson's / Schizophrenia

Urine retention / Bradycardia / Dystonic Reaction

Citalopam (Celexa)

SERT Inhibitor

Psychosis / Obsessive Compulsive / Parkinson's

SLUDGE / Serotonin Syndrome / Hypotension

Phenelzine (Nardil)

Nonselective MAO Inhibitor

Depression / Migraine Headache / Schizophrenia

Bradycardia / Hypertension / Sedation

Clobazam (Onfi)

GABA-A modulator

Analgesic / Anticonvulsant / Anxiolytic

Dystonic Reaction / Sedation / Bronchorrhea & Bronchospasm

Desvenlafaxine (Pristiq)

SNRI

Schizophrenia / Parkinson's / Antidepressant

Hypertension / Hypotension / Dystonic Reaction

Alprazolam (Xanax)

GABA-A modulator

Insomnia / Depression / Analgesic

Sedation / Constipation / Dystonic Reaction

Lisdexamfetamine (Vyvanse)

Degranulation of NE and DA vesicles

Alzheimer's / ADHD / Schizophrenia

Dystonic Reaction / Serotonin Syndrome / Tachycardia

Olanzapine (Zyprexa)

5HT2a Antagonist / D1 Antagonist

Psychosis / Antidepressant / Weight Loss

Serotonin Syndrome / Dystonic Reaction / SLUDGE

Zaleplon (Sonata)

nonbenzodiazepine GABA-A Agonist

Parkinson's / Analgesic / Insomnia

Bradycardia / Hypertension / Sedation

Selegeline (Anipryl)

MAO-B Selective Inhibition

Schizophrenia / Parkinson's / ADHD

Vomiting / Dystonic Reaction / Diarrhea & Salivation

Baclofen (Lioresal)

GABA-B Agonist

Insomnia / Anticonvulsant / Muscular Spasms

Seizures / Sedation / Tachycardia & Hypertension

Bupropion (Wellbutrin)

DAT and NET Inhibition

Depression / Insomnia / Schizophrenia

Tachycardia & Hypertension / SLUDGE / Sedation

Promethazine (Phenergan)

D1 D2 Antagonist

Analgesic / Antiemetic / Antidepressant

SLUDGE / Dystonic Reaction / Serotonin Syndrome

Paroxetine (Paxil)

SERT inhibition

ADHD / Parkinson's / Depression

Serotonin Syndrome / Dystonic Reaction / Hypotension

Ropinirole (Requip)

D2 Agonist

ADHD / Parkinson's / Depression

Nausea and Emesis / Bradycardia / Serotonin Syndrome

Explanation / Answer

DRUG

MECHANISM OF ACTION

CLINICAL INDICATION (select one)

EXPECTED ADVERSE EFFECT (select one)

Donepizil (Aricept)

Acetylcholinesterase Inhibitor

Alzheimer's

Urine retention

Citalopam (Celexa)

SERT Inhibitor

Obsessive Compulsive

Serotonin Syndrome

Phenelzine (Nardil)

Nonselective MAO Inhibitor

Depression

Hypertension

Clobazam (Onfi)

GABA-A modulator

Anticonvulsant

Sedation

Desvenlafaxine (Pristiq)

SNRI

Antidepressant

Hypertension

Alprazolam (Xanax)

GABA-A modulator

Insomnia

Constipation

Lisdexamfetamine (Vyvanse)

Degranulation of NE and DA vesicles

ADHD

Tachycardia

Olanzapine (Zyprexa)

5HT2a Antagonist / D1 Antagonist

Psychosis

Dystonic Reaction

Zaleplon (Sonata)

nonbenzodiazepine GABA-A Agonist

Insomnia

Hypertension

Selegeline (Anipryl)

MAO-B Selective Inhibition

Parkinson's

Vomiting

Baclofen (Lioresal)

GABA-B Agonist

Muscular Spasms

Seizures

Bupropion (Wellbutrin)

DAT and NET Inhibition

Depression

Tachycardia & Hypertension

Promethazine (Phenergan)

D1 D2 Antagonist

Antiemetic

Dystonic Reaction

Paroxetine (Paxil)

SERT inhibition

Depression

Serotonin Syndrome

Ropinirole (Requip)

D2 Agonist

Parkinson's

Serotonin Syndrome

DRUG

MECHANISM OF ACTION

CLINICAL INDICATION (select one)

EXPECTED ADVERSE EFFECT (select one)

Donepizil (Aricept)

Acetylcholinesterase Inhibitor

Alzheimer's

Urine retention

Citalopam (Celexa)

SERT Inhibitor

Obsessive Compulsive

Serotonin Syndrome

Phenelzine (Nardil)

Nonselective MAO Inhibitor

Depression

Hypertension

Clobazam (Onfi)

GABA-A modulator

Anticonvulsant

Sedation

Desvenlafaxine (Pristiq)

SNRI

Antidepressant

Hypertension

Alprazolam (Xanax)

GABA-A modulator

Insomnia

Constipation

Lisdexamfetamine (Vyvanse)

Degranulation of NE and DA vesicles

ADHD

Tachycardia

Olanzapine (Zyprexa)

5HT2a Antagonist / D1 Antagonist

Psychosis

Dystonic Reaction

Zaleplon (Sonata)

nonbenzodiazepine GABA-A Agonist

Insomnia

Hypertension

Selegeline (Anipryl)

MAO-B Selective Inhibition

Parkinson's

Vomiting

Baclofen (Lioresal)

GABA-B Agonist

Muscular Spasms

Seizures

Bupropion (Wellbutrin)

DAT and NET Inhibition

Depression

Tachycardia & Hypertension

Promethazine (Phenergan)

D1 D2 Antagonist

Antiemetic

Dystonic Reaction

Paroxetine (Paxil)

SERT inhibition

Depression

Serotonin Syndrome

Ropinirole (Requip)

D2 Agonist

Parkinson's

Serotonin Syndrome

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